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Catalysis

Working Paper

Automated Flow Synthesis of Artificial Heme Enzymes for Enantioselective Biocatalysis

Giulio Fittolani, Dennis A. Kutateladze, Andrei Loas, Stephen L. Buchwald, Bradley L. Pentelute

Version 1 posted 13 June 2024

840

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Organic Chemistry

Working Paper

Room-Temperature Cu-Catalyzed Etherification of Aryl Bromides

Michael Strauss, Megan Greaves, Seoung-Tae Kim, Christiana Teijaro, Michael Schmidt, Paul Scola, Stephen Buchwald

Version 1 posted 09 January 2024

1,128

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Biological and Medicinal Chemistry

Working Paper

Electrophile Scanning Reveals Reactivity Hotspots for the Design of Covalent Peptide Binders

Nathalie M. Grob, Clint Remarcik, Simon L. Rössler, Jeffrey Y. K. Wong, John C. K. Wang, Jason Tao, Corey L. Smith, Andrei Loas, Stephen L. Buchwald, Dan L. Eaton, Magdalena Preciado López, Bradley L. Pentelute

Version 1 posted 19 June 2023

1,176

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Biological and Medicinal Chemistry

Working Paper

Site-Specific Antibody Prodrugs via S-Arylation: A Bioconjugation Approach Toward Masked Tyrosine Analogues

Jason Tao, Heemal H. Dhanjee, Michael W. Gribble Jr., Veronika Kottisch, Jacob Rodriguez, Joseph S. Brown, Holly Schmidt, Juhi Juneja, Fabienne Denhez, Peter Lee, Daša Lipovšek, Stanley Krystek, Yihong Zhang, Patrick Bousquet, Yong Zhang, Bradley L. Pentelute, Stephen L. Buchwald

Version 1 posted 22 December 2023

509

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Organic Chemistry

Working Paper

Pd-Catalyzed C–N Coupling Reactions Facilitated by Organic Bases: Mechanistic Investigation Leads to Enhanced Reactivity in the Arylation of Weakly Binding Amines

Joseph Dennis, Nicholas White, Richard Liu, Stephen L. Buchwald

Version 1 posted 10 January 2019

2,104

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Catalysis

Working Paper

The Quest for the Ideal Base: Rational Design of a Nickel Precatalyst Enables Mild, Homogeneous C–N Cross-Coupling

Richard Liu, Joseph Dennis, Stephen L. Buchwald

Version 1 posted 17 January 2020

1,092

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Organic Chemistry

Working Paper

Monophosphine Ligands Promote Pd-Catalyzed C–S Cross-Coupling Reactions at Room Temperature with Soluble Bases

Jessica Xu, Richard Liu, Charles Yeung, Stephen L. Buchwald

Version 1 posted 19 April 2019

768

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Organic Chemistry

Working Paper

CuH-Catalyzed Enantioselective Ketone Allylation with 1,3-Dienes: Scope, Mechanism, and Applications

Chengxi Li, Richard Liu, Luke T. Jesikiewicz, Yang Yang, Peng Liu, Stephen L. Buchwald

Version 1 posted 14 December 2018

930

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Organic Chemistry

Working Paper

Copper Hydride-Catalyzed Enantioselective Synthesis of Axially Chiral 1,3-Disubstituted Allenes

Liela Bayeh, Stephen L. Buchwald

Version 1 posted 24 July 2019

856

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Catalysis

Working Paper

Synthesis of Pyrroles Through the CuH-Catalyzed Coupling of Enynes and Nitriles

Yujing Zhou, Lin Zhou, Luke T. Jesikiewicz, Peng Liu, Stephen L. Buchwald

Version 1 posted 16 April 2020

513

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26 results in Stephen Buchwald in Authors: Stephen Buchwald

Automated Flow Synthesis of Artificial Heme Enzymes for Enantioselective Biocatalysis

Room-Temperature Cu-Catalyzed Etherification of Aryl Bromides

Electrophile Scanning Reveals Reactivity Hotspots for the Design of Covalent Peptide Binders

Site-Specific Antibody Prodrugs via S-Arylation: A Bioconjugation Approach Toward Masked Tyrosine Analogues

Pd-Catalyzed C–N Coupling Reactions Facilitated by Organic Bases: Mechanistic Investigation Leads to Enhanced Reactivity in the Arylation of Weakly Binding Amines

The Quest for the Ideal Base: Rational Design of a Nickel Precatalyst Enables Mild, Homogeneous C–N Cross-Coupling

Monophosphine Ligands Promote Pd-Catalyzed C–S Cross-Coupling Reactions at Room Temperature with Soluble Bases

CuH-Catalyzed Enantioselective Ketone Allylation with 1,3-Dienes: Scope, Mechanism, and Applications

Copper Hydride-Catalyzed Enantioselective Synthesis of Axially Chiral 1,3-Disubstituted Allenes

Synthesis of Pyrroles Through the CuH-Catalyzed Coupling of Enynes and Nitriles

26 results in Authors: Stephen Buchwald