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Catalysis

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An Alkyne Linchpin Strategy for Drug:Pharmacophore Conjugation: Experimental and Computational Realization of a meta-Selective Inverse Sonogashira Coupling

Sandeep Porey, Xinglong Zhang, Suman Bhowmick, Vikas Kumar Singh, Srimanta Guin, Robert Paton, Debabrata Maiti

Version 1 posted 18 September 2019

1,070

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Organic Chemistry

Working Paper

A Practical and General Approach to the Late-Stage Functionalization of Complex Sulfonamides

Patrick Fier, Kevin M. Maloney

Version 1 posted 07 January 2019

1,185

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Organic Chemistry

Working Paper

Catalysis-Enabled Access to Cryptic Geldanamycin Oxides

Margaret J. Hilton, Christopher Brackett, Brandon Q. Mercado, Brian S. J. Blagg, Scott Miller

Version 1 posted 09 January 2020

550

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Catalysis

Working Paper

Combined Photoredox and Carbene Catalysis for the Synthesis of Ketones from Carboxylic Acids

Anna Davies, keegan fitzpatrick, Rick Betori, Karl Scheidt

Version 1 posted 13 January 2020

1,106

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Organic Chemistry

Working Paper

Sulfenylnitrene-Mediated Nitrogen-Atom Insertion into Pyrroles, Indoles, and Imidazoles

Bidhan Ghosh, Prakash Kafle, Rishav Mukherjee, Randall Welles, Deacon Herndon, Kenneth Nicholas, Yihan Shao, Indrajeet Sharma

Version 2 posted 26 September 2024

2,102

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Organic Chemistry

Working Paper

A modular flow platform enables selective and fast SuFEx ligation of small molecules, peptides, and proteins

Miguel Bernus, Daniele Mazzarella, Jelena Stanic, Ziran Zhai, Alejandro Yeste Vazquez, Omar Boutureira, Andrea Gargano, Tom Grossmann, Timothy Noel

Version 1 posted 26 May 2023

1,058

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Organic Chemistry

Working Paper

Visible Light Promoted Functionalisation of Carbon-Carbon Sigma Bonds

Jeremy Nugent, Carlos Arroniz, Bethany Shire, Alistair J. Sterling, Helena D. Pickford, Marie L. J. Wong, Steven J. Mansfield, Dimitri F. J. Caputo, Benjamin Owen, James J. Mousseau, Fernanda Duarte, Edward Anderson

Version 1 posted 08 April 2019

1,900

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Catalysis

Working Paper

Bringing Biocatalysis into the Deuteration Toolbox

Jack Rowbotham, Oliver Lenz, Holly Reeve, Kylie Vincent

Version 1 posted 12 April 2019

1,242

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1

Citations

Organic Chemistry

Working Paper

Asymmetric Total Synthesis of C9’-epi-Sinefungin

Ludovic Decultot, Rocco L. Policarpo, Brandon Wright, Danny Huang, Matthew Shair

Version 1 posted 19 May 2020

654

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2

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Organic Chemistry

Working Paper

Predictive Minisci and P450 Late Stage Functionalization with Transfer Learning

Emma King-Smith, Felix A. Faber, Usa Reilly, Anton V. Sinitskiy, Qingyi Yang, Bo Liu, Dennis Hyek, Alpha A. Lee

Version 3 posted 06 September 2023

1,167

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13 results in Late Stage Functionalization in Keywords: Late Stage Functionalization

An Alkyne Linchpin Strategy for Drug:Pharmacophore Conjugation: Experimental and Computational Realization of a meta-Selective Inverse Sonogashira Coupling

A Practical and General Approach to the Late-Stage Functionalization of Complex Sulfonamides

Catalysis-Enabled Access to Cryptic Geldanamycin Oxides

Combined Photoredox and Carbene Catalysis for the Synthesis of Ketones from Carboxylic Acids

Sulfenylnitrene-Mediated Nitrogen-Atom Insertion into Pyrroles, Indoles, and Imidazoles

A modular flow platform enables selective and fast SuFEx ligation of small molecules, peptides, and proteins

Visible Light Promoted Functionalisation of Carbon-Carbon Sigma Bonds

Bringing Biocatalysis into the Deuteration Toolbox

Asymmetric Total Synthesis of C9’-epi-Sinefungin

Predictive Minisci and P450 Late Stage Functionalization with Transfer Learning

13 results in Keywords: Late Stage Functionalization