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Biological and Medicinal Chemistry

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Materials Chemistry

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Targeted Therapy

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5 results in Keywords: Targeted Therapy

Biological and Medicinal Chemistry

Novel Inhibitors of Eukaryotic Elongation Factor 2 Kinase: In Silico, Synthesis, and in Vitro Studies

Ferah CÖMERT ÖNDER, Serdar DURDAĞI, Nermin Kahraman, Tuğçe Nur Uslu, Hakan Kandemir, Esen Bellur Atici, Bülent ÖZPOLAT, Mehmet AY

Version 1 posted 02 December 2020

479

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Biological and Medicinal Chemistry

Pitfalls and considerations in determining the potency and mutant selectivity of covalent epidermal growth factor receptor inhibitors

Kristopher W Hoyt, Daniel A Urul, Blessing C Ogboo, Florian Wittlinger, Stefan A Laufer, Erik M Schaefer, Earl W May, David E Heppner

Version 1 posted 24 August 2023

403

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Materials Chemistry

A Hydrogen-Bonded Organic Framework Equipped with a Molecular Nano-Valve

Sara Ghazal, Sarah Tabbalat, Felipe Gandara, Ala'a Al-Ghourani, Samah Abusulieh, Mahmoud Abdellatief, Suhair Sunoqrot, Kyle Cordova

Version 1 posted 16 August 2023

245

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Biological and Medicinal Chemistry

Design of BET Inhibitor Prodrugs with Superior Efficacy and Devoid of Systemic Toxicities

Farrukh Vohidov, Jannik N. Andersen, Kyriakos D. Economides, Michail V. Shipitsin, Olga Burenkova, James C. Ackley, Bhavatarini Vangamudi, Nolan M. Gallagher, Peyton Shieh, Matthew R. Golder, Jenny Liu, William K. Dahlberg, Hung V.-T. Nguyen, Deborah J. C. Ehrlich, Julie Kim, Sung Jin Huh, Allison M. Neenan, Joelle Baddour, Sattanathan Paramasivan, Elisa de Stanchina, Gaurab KC, David J. Turnquist, Jennifer K. Saucier-Sawyer, Paul W. Kopesky, Samantha W. Brady, Michael J. Jessel, Lawrence A. Reiter, Donald E. Chickering, Jeremiah Johnson, Peter Blume-Jensen

Version 1 posted 17 November 2020

753

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Biological and Medicinal Chemistry

Bioreducible Pro-drug Inhibitors of Enolase

Victoria Yan, Kristine Yang, Elliot Ballato, Kenisha Arthur, Dimitra Georgiou, Florian Muller

Version 1 posted 26 March 2020

518

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2

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