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Biological and Medicinal Chemistry

Working Paper

Deconstructing the potency and cell-line selectivity of membranolytic anticancer peptides

Cristina Martínez-Hernández, Mariana del Carmen Aguilera-Puga, Fabien Plisson

Version 1 posted 25 January 2023

71

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Materials Chemistry

Working Paper

Radiotherapy Enhancement by Ti3C2Tx MXenes

Monika Zimmermann, Lukas R.H. Gerken, Shianlin Wee, Vera M. Kissling, Anna Lena Neuer, Elena Tsolaki, Alexander Gogos, Maria R. Lukatskaya, Inge K. Herrmann

Version 1 posted 30 March 2023

158

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Biological and Medicinal Chemistry

Working Paper

A prodrug activated by H2O2 and mitochondrial hydroxide: an improvement of cancer cells versus neutrophils selectivity

Insa Klemt, Viktor Reshetnikov, Subrata Dutta, Galyna Bila, Rostyslav Bilyy, Itziar Cossío Cuartero, Andrés Hidalgo, Adrian Wünsche, Maximilian Böhm, Marit Wondrak, Leoni Kunz-Schughart, Rainer Tietze, Frank Beierlein, Petra Imhof, Sabrina Gensberger-Reigl, Monika Pischetsrieder, Marlies Körber, Tina Jost, Andriy Mokhir

Version 2 posted 27 September 2023

281

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Inorganic Chemistry

Working Paper

Polymeric Encapsulation of a Ruthenium(II) Polypyridyl Complex: From Synthesis to in vivo Studies against High-Grade Epithelial Ovarian Cancer

Gilles Gasser, Joao Antonio, Albert Gandioso, Fariba Nemati, Nancy Soliman, Robin Vinck, Fan Sun, Carine Robert, Pierre Burckel, Didier Decaudin, Christophe Thomas

Version 1 posted 13 October 2022

186

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Biological and Medicinal Chemistry

Working Paper

Identification of the FDA-Approved Drug Pyrvinium as a Novel Inhibitor of PD-1/PD-L1 Interaction

Elena Fattakhova, Jeremy Hofer, Juliette DiFlumeri, Madison Cobb, Timothy Dando, Zachary Romisher, Justin Wellington, Michael Oravic, Madison Radnoff, Sachin Patil

Version 1 posted 19 April 2021

349

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Biological and Medicinal Chemistry

Working Paper

Tuaimenal A, a Meroterpene from the Irish Deep-Sea Soft Coral Duva florida, Displays Inhibition of the SARS-CoV-2 3CLpro Enzyme.

Nicole E. Avalon, Jordan Nafie, Carolina De Marco Verissimo, Luke C. Warrensford, Sarah G. Dietrick, Amanda R. Pittman, Ryan M. Young, Fiona L. Kearns, Tracess Smalley, Jennifer M. Binning, John P. Dalton, Mark P. Johnson, H. Lee Woodcock, A. Louise Allcock, Bill J. Baker

Version 3 posted 12 May 2022

905

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Biological and Medicinal Chemistry

Working Paper

Computer-aided design, synthesis, and biological evaluation of [4.3.0] bicyclic prolyl oligopeptidase and fibroblast activation protein-α dual inhibitors

Nicolas Moitessier, Jessica Plescia, Damien Hedou, Maud Pousse, Anne Labarre, Caroline Dufresne, Anthony Mittermaier

Version 1 posted 30 August 2021

378

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Biological and Medicinal Chemistry

Working Paper

Thiamine Analogues as Tools to Study Pyruvate Dehydrogenase in Cancer: Biochemical, Computational and Cellular Analyses

Finian James Leeper, Alex Chan, Terence Ho, Daniel Parle

Version 1 posted 19 September 2022

184

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1

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Inorganic Chemistry

Working Paper

Bis[Pyrrolyl Ru(II)] Triads: a New Class of Photosensitizers for Metal-Organic Photodynamic Therapy

Deborah A. Smithen, Susan Monro, Mitch Pinto, John A. Roque III, Roberto M. Diaz-Rodriguez, Huimin Yin, Colin G. Cameron, Alison Thompson, Sherri A. McFarland

Version 1 posted 25 August 2020

363

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Organic Chemistry

Working Paper

Cellular Fucosylation Inhibitors Based on Fluorinated Fucose-1-Phosphates

Johan Pijnenborg, eline visser, Marek Noga, Emiel Rossing, Raisa Veizaj, Dirk J. Lefeber, Christian Büll, Thomas Boltje

Version 1 posted 10 November 2020

399

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Refine Search

66 results in Cancer in Keywords: Cancer

Deconstructing the potency and cell-line selectivity of membranolytic anticancer peptides

Radiotherapy Enhancement by Ti3C2Tx MXenes

A prodrug activated by H2O2 and mitochondrial hydroxide: an improvement of cancer cells versus neutrophils selectivity

Polymeric Encapsulation of a Ruthenium(II) Polypyridyl Complex: From Synthesis to in vivo Studies against High-Grade Epithelial Ovarian Cancer

Identification of the FDA-Approved Drug Pyrvinium as a Novel Inhibitor of PD-1/PD-L1 Interaction

Tuaimenal A, a Meroterpene from the Irish Deep-Sea Soft Coral Duva florida, Displays Inhibition of the SARS-CoV-2 3CLpro Enzyme.

Computer-aided design, synthesis, and biological evaluation of [4.3.0] bicyclic prolyl oligopeptidase and fibroblast activation protein-α dual inhibitors

Thiamine Analogues as Tools to Study Pyruvate Dehydrogenase in Cancer: Biochemical, Computational and Cellular Analyses

Bis[Pyrrolyl Ru(II)] Triads: a New Class of Photosensitizers for Metal-Organic Photodynamic Therapy

Cellular Fucosylation Inhibitors Based on Fluorinated Fucose-1-Phosphates

66 results in Keywords: Cancer