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10 results in Keywords: Acylation

Biological and Medicinal Chemistry

Working Paper

Cationic, Aromatic Acyl Donors for Directing Protein Acylation Using non-Covalent Interactions

Nicholas Kuehl, Hieu Pham, Joseph Ault, Michael Taylor

Version 1 posted 30 April 2024

400

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Catalysis

Working Paper

Nickel-Catalyzed Acylation of Aryl Bromides with Acyl Imidazoles

Junming Zhuo, Yong Zhang, Zijian Li, Chao Li

Version 1 posted 12 July 2019

1,301

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Catalysis

Working Paper

Mild Organic Base-Catalyzed Primary Alcohol-Selective Aroylation Reaction Using N-Aroylcarbazoles for Underexplored Prodrugs

Yasuaki Morita, Bubwoong Kang, Rubi Nakashima, Yuki Shimizu, Asumi Sakai, Maiko Moriguchi, Yoko Yasuno, Tetsuya Satoh, Tetsuro Shinada, Masaki Kuse

Version 1 posted 09 June 2020

713

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Organic Chemistry

Working Paper

Post Glycosylation Diversification (PGD): An Approach for Assembling Collections of Glycosylated Small Molecules

Zachary Cannone, Ala Shaqra, Chris Lorenc, Liza Henowitz, Santosh Keshipeddy, Victoria Robinson, Adam Zweifach, Dennis Wright, Mark Peczuh

Version 1 posted 21 September 2018

533

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Organic Chemistry

Working Paper

Progress Towards a Large-Scale Synthesis of Molnupiravir (MK-4482, EIDD-2801) from Cytidine

Grace P. Ahlqvist, Catherine P. McGeough, Chris Senanayake, Joseph D. Armstrong, Ajay Yadaw, Sarabindu Roy, Saeed Ahmad, David R. Snead, Tim Jamison

Version 1 posted 16 February 2021

1,680

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Citations

Organic Chemistry

Working Paper

N-Acyl-1,2,3-triazoles - key intermediates in denitrogenative transformations

Vladimir Motornov, Radek Pohl, Blanka Klepetářová, Petr Beier

Version 1 posted 08 March 2023

285

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Theoretical and Computational Chemistry

Working Paper

Unraveling the SARS-CoV-2 Main Protease Mechanism Using Multiscale DFT/MM Methods

Carlos A. Ramos-Guzmán, J. Javier Ruiz-Pernía, Iñaki Tuñón

Version 2 posted 07 July 2020

1,118

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Citations

Catalysis

Working Paper

Thioester Mediated Biocatalytic Amide Bond Synthesis with In Situ Thiol Recycling

Christian Schnepel, Laura Rodriguez-Perez, Yuqi Yu, Antonio Angelastro, Rachel S. Heath, Max Lubberink, Francesco Falcioni, Keith Mulholland, Martin A. Hayes, Nicholas J. Turner, Sabine L. Flitsch

Version 3 posted 05 May 2022

1,718

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Catalysis

Working Paper

Isothiourea-Catalysed Acylative Dynamic Kinetic Resolution of Tetra-substituted Morpholinone and Benzoxazinone Lactols

Haoxiang Zhu, Alejandro Manchado, Abdikani Omar Farah, Aidan McKay, David Cordes, Paul Ha-Yeon Cheong, Kevin Kasten, Andrew Smith

Version 1 posted 31 January 2024

342

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Organic Chemistry

Working Paper

Enantioselective Synthesis of Tetra-substituted 3-Hydroxyphthalide Esters by Isothiourea-Catalysed Acylative Dynamic Kinetic Resolution

Shubham Agrawal, Pankaj Majhi, Alister Goodfellow, Raj Tak, David Cordes, Aidan McKay, Kevin Kasten, Michael Buehl, Andrew Smith

Version 1 posted 31 January 2024

361

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10 results in Acylation in Keywords: Acylation

Cationic, Aromatic Acyl Donors for Directing Protein Acylation Using non-Covalent Interactions

Nickel-Catalyzed Acylation of Aryl Bromides with Acyl Imidazoles

Mild Organic Base-Catalyzed Primary Alcohol-Selective Aroylation Reaction Using N-Aroylcarbazoles for Underexplored Prodrugs

Post Glycosylation Diversification (PGD): An Approach for Assembling Collections of Glycosylated Small Molecules

Progress Towards a Large-Scale Synthesis of Molnupiravir (MK-4482, EIDD-2801) from Cytidine

N-Acyl-1,2,3-triazoles - key intermediates in denitrogenative transformations

Unraveling the SARS-CoV-2 Main Protease Mechanism Using Multiscale DFT/MM Methods

Thioester Mediated Biocatalytic Amide Bond Synthesis with In Situ Thiol Recycling

Isothiourea-Catalysed Acylative Dynamic Kinetic Resolution of Tetra-substituted Morpholinone and Benzoxazinone Lactols

Enantioselective Synthesis of Tetra-substituted 3-Hydroxyphthalide Esters by Isothiourea-Catalysed Acylative Dynamic Kinetic Resolution

10 results in Keywords: Acylation