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Deep Alanine Scanning Reveals Potent Multi-alanine-substituted Protein–protein Interaction Inhibitors

Xiyun Ye, Yen-Chun Lee, Zachary P. Gates, Yingjie Ling, Jennifer Mortensen, Fan-Shen Yang, Yu-Shan Lin, Bradley Pentelute

Version 1 posted 21 January 2021

709

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1

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Organic Chemistry

Working Paper

Automated Fast-Flow Synthesis of C9orf72 Dipeptide Repeat Proteins

Kohei Sato, Charlotte E. Farquhar, Bradley Pentelute

Version 1 posted 06 March 2023

346

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Biological and Medicinal Chemistry

Working Paper

Reversibly reactive affinity selection mass spectrometry enables maturation of covalent peptides

Peiyuan Zhang, Xiyun Ye, John C.K. Wang, Hannah T. Baddock, Zena Jensvold, Ian Foe, Andrei Loas, Dan L. Eaton, Qi Hao, Aaron H. Nile, Bradley L. Pentelute

Version 1 posted 22 December 2023

467

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Biological and Medicinal Chemistry

Working Paper

Linearizable Macrocyclic Peptide Libraries for Affinity Selection-Mass Spectrometry

Michael A. Lee, Joseph S. Brown, Charlotte E. Farquhar, Andrei Loas, Bradley L. Pentelute

Version 1 posted 05 February 2024

447

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Biological and Medicinal Chemistry

Working Paper

Electrophile Scanning Reveals Reactivity Hotspots for the Design of Covalent Peptide Binders

Nathalie M. Grob, Clint Remarcik, Simon L. Rössler, Jeffrey Y. K. Wong, John C. K. Wang, Jason Tao, Corey L. Smith, Andrei Loas, Stephen L. Buchwald, Dan L. Eaton, Magdalena Preciado López, Bradley L. Pentelute

Version 1 posted 19 June 2023

1,095

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1

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Biological and Medicinal Chemistry

Working Paper

Abiotic peptides for the encoding of small molecule synthesis

Simon L. Rössler, Nathalie M. Grob, Stephen L. Buchwald, Bradley L. Pentelute

Version 1 posted 27 September 2022

1,531

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Biological and Medicinal Chemistry

Working Paper

Rapid Production of Native and Mirror-Image Tumor Necrosis Factor-α through the Synergy of Automated Flow Peptide Synthesis and Native Chemical Ligation

Ahmet Yesilcimen, Alex J. Callahan, Tara L. Travaline, Satish Gandhesiri, Olena S. Tokareva, Andrei Loas, John H. McGee, Bradley L. Pentelute

Version 1 posted 02 February 2024

309

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Biological and Medicinal Chemistry

Working Paper

Site-Specific Antibody Prodrugs via S-Arylation: A Bioconjugation Approach Toward Masked Tyrosine Analogues

Jason Tao, Heemal H. Dhanjee, Michael W. Gribble Jr., Veronika Kottisch, Jacob Rodriguez, Joseph S. Brown, Holly Schmidt, Juhi Juneja, Fabienne Denhez, Peter Lee, Daša Lipovšek, Stanley Krystek, Yihong Zhang, Patrick Bousquet, Yong Zhang, Bradley L. Pentelute, Stephen L. Buchwald

Version 1 posted 22 December 2023

433

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Organic Chemistry

Working Paper

Same Day Access to Proteins Enabled by Folding Selections

Alex J. Callahan, Aurélie Rondon, Lia Lozano Salazar, Satish Gandhesiri, Jacob Rodriguez, Andrei Loas, Bradley Pentelute

Version 1 posted 17 April 2023

442

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Theoretical and Computational Chemistry

Working Paper

Unsupervised machine learning leads to an abiotic picomolar peptide ligand

Joseph S. Brown, Somesh Mohapatra, Michael A. Lee, Roman Misteli, Yitong Tseo, Nathalie M. Grob, Anthony J. Quartararo, Andrei Loas, Rafael Gomez-Bombarelli, Bradley L. Pentelute

Version 1 posted 24 May 2023

906

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18 results in Bradley Pentelute in Authors: Bradley Pentelute

Deep Alanine Scanning Reveals Potent Multi-alanine-substituted Protein–protein Interaction Inhibitors

Automated Fast-Flow Synthesis of C9orf72 Dipeptide Repeat Proteins

Reversibly reactive affinity selection mass spectrometry enables maturation of covalent peptides

Linearizable Macrocyclic Peptide Libraries for Affinity Selection-Mass Spectrometry

Electrophile Scanning Reveals Reactivity Hotspots for the Design of Covalent Peptide Binders

Abiotic peptides for the encoding of small molecule synthesis

Rapid Production of Native and Mirror-Image Tumor Necrosis Factor-α through the Synergy of Automated Flow Peptide Synthesis and Native Chemical Ligation

Site-Specific Antibody Prodrugs via S-Arylation: A Bioconjugation Approach Toward Masked Tyrosine Analogues

Same Day Access to Proteins Enabled by Folding Selections

Unsupervised machine learning leads to an abiotic picomolar peptide ligand

18 results in Authors: Bradley Pentelute