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Resin-assisted synthesis of a neopentyl 211At-labeled activated ester possessing a triazole spacer and its application to the synthesis of in vivo stable 211At-labeled antibodies.

Masatoshi Tada, Yuta Kaizuka, Kento Kannaka, Hiroyuki Suzuki, Taiki Joho, Kazuhiro Takahashi, Tomoya Uehara, Hiroshi Tanaka

Version 1 posted 02 April 2024

147

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Biological and Medicinal Chemistry

Working Paper

Imaging poly(ADP-ribose) polymerase-1 (PARP1) in vivo with 18F-labeled brain penetrant positron emission tomography (PET) ligand

Xin Zhou, Jiahui Chen, Jimmy S. Patel, Wenqing Ran, Yinlong Li, Richard S. Van, Mostafa M. H. Ibrahim, Chunyu Zhao, Yabiao Gao, Jian Rong, Ahmad F. Chaudhary, Guocong Li, Junqi Hu, April T. Davenport, James D. Daunais, Yihan Shao, Chongzhao Ran, Thomas L. Collier, Ahmed Haider, David M. Schuster, Allan Levey, Lu Wang, Gabriel Corfas, Steven H. Liang

Version 2 posted 08 February 2024

544

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Biological and Medicinal Chemistry

Working Paper

Development of the First Aliphatic 18F-Labeled Tetrazine Suitable for Pretargeted PET Imaging – Expanding the Bioorthogonal Tool Box

Umberto Maria Battisti, Klas Bratteby, Jesper Tranekjær Jørgensen, Lars Hvass, Vladimir Shalgunov, Hannes Mikula, Andreas Kjaer, Matthias Herth

Version 1 posted 19 April 2021

419

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Biological and Medicinal Chemistry

Working Paper

Direct Aromatic 18F-Labeling of Highly Reactive Tetrazines for Pretargeted Bioorthogonal PET Imaging

Rocio Garcia-Vazquez, Umberto Maria Battisti, Jesper Tranekjær Jørgensen, Vladimir Shalgunov, Lars Hvass, Daniel L. Stares, Ida Nymann Petersen, François Crestey, Andreas Löffler, Dennis Svatunek, Jesper Langgaard Kristensen, Hannes Mikula, Andreas Kjaer, Matthias Herth

Version 1 posted 22 February 2021

579

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Organic Chemistry

Working Paper

Pretargeted Imaging Beyond the Blood-Brain-Barrier

Vladimir Shalgunov, Sara Lopes van den Broek, Ida Vang Andersen, Rocío García Vázquez, Nakul Raval, Mikael Palner, Yuki Mori, Gabriela Schäfer, Hannes Mikula, Natalie Beschorner, Maiken Nedergaard, Stina Syvänen, Matthias Barz, Gitte Moos Knudsen, Umberto Maria Battisti, Matthias Herth

Version 2 posted 13 April 2022

610

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3

Citations

Biological and Medicinal Chemistry

Working Paper

18F-Fluorination of 2-methyl-6-nitrobenzenesulfonate ester and its application to the synthesis of a 18F-labeled amino acid.

Shogo Iida, Tetsuro Tago, Masatoshi Tada, Jun Toyohara, Hiroshi Tanaka

Version 3 posted 07 August 2023

265

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Organic Chemistry

Working Paper

Insights into Elution of Anion Exchange Cartridges: Opening the Path towards Aliphatic 18F-Radiolabeling of Base-Sensitive Tracers

Klas Bratteby, Vladimir Shalgunov, Umberto Maria Battisti, Ida Nymann Petersen, Sara Lopes van den Broek, Tomas G Ohlsson, Nic Gillings, Maria Erlandsson, Matthias Herth

Version 1 posted 18 March 2021

653

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1

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Biological and Medicinal Chemistry

Working Paper

[18F]SuFEx Click Chemistry Enabled Ultrafast Late-stage Radiosynthesis

Qinheng Zheng, Hongtao Xu, Hua Wang, Wen-Ge Han Du, Nan Wang, Huan Xiong, Yuang Gu, Louis Noodleman, Guang Yang, K. Barry Sharpless, Peng Wu

Version 2 posted 11 August 2020

1,994

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1

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Inorganic Chemistry

Working Paper

Scalable 18F Processing Conditions for Copper-Mediated Radiofluorination Chemistry Facilitate "Design of Experiments" (DoE) Optimization Studies and Afford an Improved Synthesis of [18F]Olaparib.

Gregory D. Bowden, Nantanat Chailanggar, Bernd J. Pichler, Andreas Maurer

Version 1 posted 07 May 2021

673

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1

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Organic Chemistry

Working Paper

Lipophilicity and Click Reactivity Determine the Performance of Bioorthogonal Tetrazine Tools in Pretargeted in Vivo Chemistry

Johanna Stéen, Jesper Tranekjær Jørgensen, Denk Christoph, Umberto Maria Battisti, Kamilla Nørregaard, Patricia Edem, Klas Bratteby, Vladimir Shalgunov, Wilkovitsch Martin, Dennis Svatunek, Christian Bernard Matthijs Poulie, Lars Hvass, Marina Simon, Wanek Thomas, Raffaella Rossin, Marc Robillard, Jesper Langgaard Kristensen, Hannes Mikula, Andreas Kjaer, Matthias Herth

Version 1 posted 24 December 2020

450

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1

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Refine Search

11 results in fluorine-18 in Keywords: fluorine-18

Resin-assisted synthesis of a neopentyl 211At-labeled activated ester possessing a triazole spacer and its application to the synthesis of in vivo stable 211At-labeled antibodies.

Imaging poly(ADP-ribose) polymerase-1 (PARP1) in vivo with 18F-labeled brain penetrant positron emission tomography (PET) ligand

Development of the First Aliphatic 18F-Labeled Tetrazine Suitable for Pretargeted PET Imaging – Expanding the Bioorthogonal Tool Box

Direct Aromatic 18F-Labeling of Highly Reactive Tetrazines for Pretargeted Bioorthogonal PET Imaging

Pretargeted Imaging Beyond the Blood-Brain-Barrier

18F-Fluorination of 2-methyl-6-nitrobenzenesulfonate ester and its application to the synthesis of a 18F-labeled amino acid.

Insights into Elution of Anion Exchange Cartridges: Opening the Path towards Aliphatic 18F-Radiolabeling of Base-Sensitive Tracers

[18F]SuFEx Click Chemistry Enabled Ultrafast Late-stage Radiosynthesis

Scalable 18F Processing Conditions for Copper-Mediated Radiofluorination Chemistry Facilitate "Design of Experiments" (DoE) Optimization Studies and Afford an Improved Synthesis of [18F]Olaparib.

Lipophilicity and Click Reactivity Determine the Performance of Bioorthogonal Tetrazine Tools in Pretargeted in Vivo Chemistry

11 results in Keywords: fluorine-18