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Biological and Medicinal Chemistry

Working Paper

Peptidomimetic small-molecule inhibitors of 3CLPro activity and Spike-ACE2 interaction: towards dual-action molecules against Coronavirus infections

Filomena Tedesco, Lorenzo Calugi, Elena Lenci, Andrea Trabocchi

Version 1 posted 18 April 2022

253

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Biological and Medicinal Chemistry

Working Paper

Electrophile Scanning Reveals Reactivity Hotspots for the Design of Covalent Peptide Binders

Nathalie M. Grob, Clint Remarcik, Simon L. Rössler, Jeffrey Y. K. Wong, John C. K. Wang, Jason Tao, Corey L. Smith, Andrei Loas, Stephen L. Buchwald, Dan L. Eaton, Magdalena Preciado López, Bradley L. Pentelute

Version 1 posted 19 June 2023

1,176

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1

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Biological and Medicinal Chemistry

Working Paper

Constrained TACC3 peptidomimetics for a non-canonical protein-protein interface elucidate allosteric communication in Aurora-A Kinase

Diana Gimenez, Martin Walko, Jennifer Miles, Megan Wright, Richard Bayliss, Wilson Andrew

Version 1 posted 09 September 2024

118

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Biological and Medicinal Chemistry

Working Paper

A Photoactivatable α5β1-Specific Integrin Ligand

Roshna Vakkeel, Aleeza Farrukh, Aranzazu del Campo

Version 1 posted 06 April 2018

833

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Biological and Medicinal Chemistry

Working Paper

Optimal Anchoring of a Urea-based Foldamer Inhibitor of ASF1 Histone Chaperone Through Backbone Plasticity

Johanne Mbianda, May Bakail, Christophe André, Gwenaëlle Moal, Marie E. Perrin, Raphaël Guerois, François Becher, Pierre Legrand, Seydou Traore, Céline Douat, Gilles GUICHARD, Francoise OCHSENBEIN

Version 1 posted 09 July 2020

413

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Biological and Medicinal Chemistry

Working Paper

From Aggregation to Inhibition: N-Amination Converts Amyloidogenic Tau Peptides into Soluble Antagonists of Cellular Seeding

Kamlesh Makwana, Matthew P. Sarnowski, Jiyuan Miao, Yu-Shan Lin, Juan Del Valle

Version 1 posted 26 April 2021

368

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Organic Chemistry

Working Paper

Metal-Binding Q-Proline Macrocycles

Justin Northrup, Jesse Wiener, Matthew Hurley, Chun-Feng David Hou, Taylor Keller, Richard Baxter, Michael J. Zdilla, Vincent Voelz, Christian Schafmeister

Version 1 posted 12 January 2021

331

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Theoretical and Computational Chemistry

Working Paper

Unsupervised machine learning leads to an abiotic picomolar peptide ligand

Joseph S. Brown, Somesh Mohapatra, Michael A. Lee, Roman Misteli, Yitong Tseo, Nathalie M. Grob, Anthony J. Quartararo, Andrei Loas, Rafael Gomez-Bombarelli, Bradley L. Pentelute

Version 1 posted 24 May 2023

1,072

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Biological and Medicinal Chemistry

Working Paper

Design and Synthesis of Novel Peptidomimetics for Cancer Immunotherapy

Ceyda Köse, Esra Uysal, Büşra Yazıcı, Zeynep Tuğay, Serap İpek Dingiş Birgül, Hamdullah Yanık, Ece Tavukcuoglu, Sevgi Gulyuz, Atilla Akdemir, Güneş Esendağlı, Özgür Yılmaz, Onur Alptürk

Version 1 posted 10 September 2020

356

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Biological and Medicinal Chemistry

Working Paper

Peptoid-Based Reprogrammable Template for Cell-Permeable Inhibitors of Protein–Protein Interactions

Yasuhiro Fukuda, Marin Yokomine, Daisuke Kuroda, Kouhei Tsumoto, Jumpei Morimoto, Shinsuke Sando

Version 1 posted 05 May 2021

321

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16 results in Peptidomimetics in Keywords: Peptidomimetics

Peptidomimetic small-molecule inhibitors of 3CLPro activity and Spike-ACE2 interaction: towards dual-action molecules against Coronavirus infections

Electrophile Scanning Reveals Reactivity Hotspots for the Design of Covalent Peptide Binders

Constrained TACC3 peptidomimetics for a non-canonical protein-protein interface elucidate allosteric communication in Aurora-A Kinase

A Photoactivatable α5β1-Specific Integrin Ligand

Optimal Anchoring of a Urea-based Foldamer Inhibitor of ASF1 Histone Chaperone Through Backbone Plasticity

From Aggregation to Inhibition: N-Amination Converts Amyloidogenic Tau Peptides into Soluble Antagonists of Cellular Seeding

Metal-Binding Q-Proline Macrocycles

Unsupervised machine learning leads to an abiotic picomolar peptide ligand

Design and Synthesis of Novel Peptidomimetics for Cancer Immunotherapy

Peptoid-Based Reprogrammable Template for Cell-Permeable Inhibitors of Protein–Protein Interactions

16 results in Keywords: Peptidomimetics