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Biological and Medicinal Chemistry

Working Paper

A Generative Deep Learning Approach for the Discovery of SARS CoV2 Protease Inhibitors

Noor Shaker, Mohamed Abou-Zleikha, Mubarak AlAmri, Youcef Mehellou

Version 1 posted 23 April 2020

1,480

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2

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Biological and Medicinal Chemistry

Working Paper

Pan-Specific and Partially Selective Dye-Labeled Peptidic Inhibitors of the Polycomb Paralog Proteins

Natalia Milosevich, James McFarlane, Michael Gignac, Janessa Li, Tyler Brown, Chelsea Wilson, Lindsay Devorkin, Caitlin Croft, Rebecca Hof, Irina Paci, Julian Lum, Fraser Hof

Version 1 posted 15 July 2019

715

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Biological and Medicinal Chemistry

Working Paper

Aryloxy Triester Phosphoramidates as Phosphoserine Biocleavable Masking Motifs

Ageo Miccoli, Binar A. Dhiani, Peter J. Thornton, Olivia A. Lambourne, Edward James, Hachemi Kadri, Youcef Mehellou

Version 1 posted 13 November 2019

496

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Organic Chemistry

Working Paper

Cellular Fucosylation Inhibitors Based on Fluorinated Fucose-1-Phosphates

Johan Pijnenborg, eline visser, Marek Noga, Emiel Rossing, Raisa Veizaj, Dirk J. Lefeber, Christian Büll, Thomas Boltje

Version 1 posted 10 November 2020

420

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Biological and Medicinal Chemistry

Working Paper

Theoretical Study of the anti-NCP Molecular Mechanism of Traditional Chinese Medicine Lianhua-Qingwen Formula (LQF)

Chenghao Ye, Meina Gao, Wangqiang Lin, Kunqian Yu, Peng Li, Guanghui Chen

Version 1 posted 23 March 2020

3,171

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2

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Biological and Medicinal Chemistry

Working Paper

Structure-based Discovery of a Series of NSD2-PWWP1 Inhibitors

Na Li, Hong Yang, Ke Liu, Liwei Zhou, Yuting Huang, Danyan Cao, Yanlian Li, Yaoliang Sun, Aisong Yu, Zhiyan Du, Feng Yu, Ying Zhang, Bingyang Wang, Meiyu Geng, Jian Li, Shilin Xu, Bing Xiong, Xun Huang, Tongchao Liu

Version 2 posted 08 December 2021

929

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Biological and Medicinal Chemistry

Working Paper

Open-chain thiamine analogues as potent inhibitors of thiamine pyrophosphate (TPP)-dependent enzymes

Alex H. Y. Chan, Terence C. S. Ho, Finian James Leeper

Version 1 posted 30 May 2023

99

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Biological and Medicinal Chemistry

Working Paper

Novel dihydropteridinone derivatives as potent and selective inhibitors of the understudied human vaccinia-related kinase 1 (VRK1)

Fernando H. de Souza Gama, Luiz Dutra, Michael Hawgood, Caio Vinícius dos Reis, Ricardo Serafim, Marcos Ferreira Jr., Bruno V. M. Teodoro, Jéssica Takarada, André Santiago, Vitor M. Almeida, Carina Gileadi, Priscila Zonzini Ramos, Anita Salmazo, Stanley Vasconcelos, Micael Cunha, Dimitrios-Ilias Ballourdas, Susanne Mueller, Stefan Knapp, Katlin Massirer, Jonathan Elkins, Opher Gileadi, Alessandra Macarello, Bennie Lemmens, Cristiano R. W. Guimarães, Hatylas Azevedo, Rafael Couñago

Version 1 posted 04 December 2023

1,009

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Biological and Medicinal Chemistry

Working Paper

On the potential pharmacophore for the structure-based inhibitor design against phosphatases

Petar M. Mitrasinovic

Version 1 posted 27 August 2024

82

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Materials Science

Working Paper

Corrosion Inhibition of AZ31-xLi (x = 4, 8, 12) Magnesium Alloys in Sodium Chloride Solutions by Aqueous Molybdate

Maria Osipenko, Andrei Paspelau, Aliaksandr Kasach, Jacek Ryl, Konrad Skowron, Janusz Adamiec, Irina Kurilo, Dzmitry Kharytonau

Version 1 posted 22 March 2024

126

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Refine Search

28 results in Inhibitor, Sucralose in Keywords: Inhibitor, Sucralose

A Generative Deep Learning Approach for the Discovery of SARS CoV2 Protease Inhibitors

Pan-Specific and Partially Selective Dye-Labeled Peptidic Inhibitors of the Polycomb Paralog Proteins

Aryloxy Triester Phosphoramidates as Phosphoserine Biocleavable Masking Motifs

Cellular Fucosylation Inhibitors Based on Fluorinated Fucose-1-Phosphates

Theoretical Study of the anti-NCP Molecular Mechanism of Traditional Chinese Medicine Lianhua-Qingwen Formula (LQF)

Structure-based Discovery of a Series of NSD2-PWWP1 Inhibitors

Open-chain thiamine analogues as potent inhibitors of thiamine pyrophosphate (TPP)-dependent enzymes

Novel dihydropteridinone derivatives as potent and selective inhibitors of the understudied human vaccinia-related kinase 1 (VRK1)

On the potential pharmacophore for the structure-based inhibitor design against phosphatases

Corrosion Inhibition of AZ31-xLi (x = 4, 8, 12) Magnesium Alloys in Sodium Chloride Solutions by Aqueous Molybdate

28 results in Keywords: Inhibitor, Sucralose