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Biological and Medicinal Chemistry

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Organic Chemistry

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BRET

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4 results in Keywords: BRET

Biological and Medicinal Chemistry

Enzyme-mediated proximity labeling for enrichment of DNA-linked ligands from DNA-encoded libraries

Bo Cai, Amol Mhetre, Casey Krusemark

Version 1 posted 05 October 2022

672

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Biological and Medicinal Chemistry

Novel Pyrazolo[3,4-c]pyridine Antagonists with Nanomolar affinity for A1 / A3 Adenosine Receptors: Binding Kinetics and Exploration of their Binding Profile Using Mutagenesis Experiments, MD simulations and TI/MD calculations

Margarita Stampelou, Anna Suchankova, Efpraxia Tzortzini, Lakshiv Dhingra, Kerry Barkan, Nikolaos Lougiakis, Panagiotis Marakos, Nikole Pouli, Graham Ladds, Antonios Kolocouris

Version 4 posted 24 November 2021

472

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Biological and Medicinal Chemistry

Synthetic Analogs of the Snail Toxin 6-Bromo-2-Mercaptotryptamine Dimer (BrMT) Reveal That Lipid Bilayer Perturbation Does Not Underlie Its Modulation of Voltage-Gated Potassium Channels

Chris Dockendorff, Disha M. Gandhi, Ian H. Kimball, Kenneth S. Eum, Radda Rusinova, Helgi I. Ingólfsson, Ruchi Kapoor, Thasin Peyear, Matthew W. Dodge, Stephen F. Martin, Richard W. Aldrich, Olaf S. Andersen, Jon T. Sack

Version 1 posted 21 February 2018

431

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Biological and Medicinal Chemistry

Comprehensive Survey of CDK Inhibitor Selectivity in Live Cells with Energy Transfer Probes

Carrow Wells, Jim Vasta, Cesear R. Corona, Jennifer Wilkinson, Chad A. Zimprich, Morgan R. Ingold, Julie E. Pickett, David Drewry, Kathryn Maria Pugh, Kilian Huber, Mei Cong, Poncho Meisenheimer, Timothy M. Willson, Matthew B. Robers

Version 1 posted 23 December 2019

1,218

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