Category:
Biological and Medicinal Chemistry
,
Working Paper
, Title:
Azapeptide-based SARS-CoV-2 Main Protease Inhibitors: Design, Synthesis, Enzyme Inhibition, Structural Determination, and Antiviral Activity
, Authors:
Philipp Flury, Jyoti Vishwakarma, Katharina Sylvester, Nobuyo Higashi-Kuwata, Agnieszka Dabrowska, Renee Delgado, Ashley Cuell, Rahul Basu, Alexander B. Taylor, Ellen Gonçalves de Oliveira, Mateus Sá Magalhães Serafim, Jingxin Qiao, Yan Chen, Shengyong Yang, Anthony J. O’Donoghue, Hiroaki Mitsuya, Michael Gütschow, Stefan A. Laufer, Christa E. Müller, Reuben S. Harris, Thanigaimalai Pillaiyar
Version 1 posted 04 June 2025
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