Abstract
1-Azaspiro[3.3]heptanes were synthesized, characterized, and validated biologically in vivo as a new generation of saturated piperidine bioisosteres.
Supplementary materials
Title
SI
Description
Supporting Information.
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Bicyclic Bioisosteres of Piperidine: Version 2.0
12 April 2023, Version 1
Working Paper
This content is a preprint and has not undergone peer review at the time of posting.
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Version History
Apr 12, 2023 Version 1
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Funding
European Research Council
101000893
Author’s competing interest statement
Authors of this work are employees of a chemical supplier Enamine.
Ethics
The author(s) declare that they have sought and gained approval from the
relevant ethics committee/IRB for this research and its publication.