Organic Chemistry

Mild and Chemoselective Phosphorylation of Alcohols Using a PSI-Reagent



An operationally simple, scalable, and chemoselective method for the direct phosphorylation of alcohols using a P(V)-approach based on the PSI-reagent platform is disclosed. The method features a broad substrate scope of utility in both simple and complex settings and provides access to valuable phosphorylated alcohols that would be otherwise difficult to access.


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Supplementary material

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Supporting information
copies of spectra, characterization, and procedures