Organic Chemistry

Facile Synthesis of a Diverse Library of Mono-3-substituted β-Cyclodextrin Analogues



We have described simple, high-yield, protocols, which require only commonly accessible equipment, to synthesize a wide range of β-CD derivatives mono-substituted at the secondary face. These derivatives may be useful in their own right, and they are also scaffolds for further modification, and examples of the far broader array of derivatives that may be accessed by these procedures.

Version notes

We have added four more cyclodextrin analogues to the paper.


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Supplementary material

Thumbnail image of Gilson_CD_synthesis_SI.pdf
Gilson CD synthesis SI
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CD synthesis SI 2
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Gilson CD synthesis