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Facile Synthesis of a Diverse Library of Mono-3-substituted β-Cyclodextrin Analogues

revised on 26.07.2018, 16:44 and posted on 26.07.2018, 16:57 by Kathryn Kellett, Brendan M. Duggan, Michael Gilson
We have described simple, high-yield, protocols, which require only commonly accessible equipment, to synthesize a wide range of β-CD derivatives mono-substituted at the secondary face. These derivatives may be useful in their own right, and they are also scaffolds for further modification, and examples of the far broader array of derivatives that may be accessed by these procedures.


Email Address of Submitting Author


University of California, San Diego


United States of America

ORCID For Submitting Author


Declaration of Conflict of Interest

M.K.G. has an equity interest in, and is a cofounder and scientific advisor of VeraChem LLC.

Version Notes

We have added four more cyclodextrin analogues to the paper.