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Biological and Medicinal Chemistry

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Organic Chemistry

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G protein-coupled receptor

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5 results in Keywords: G protein-coupled receptor

Biological and Medicinal Chemistry

Discovery of 2-aminopyrimidines as potent agonists for the bitter taste receptor TAS2R14

Lukas Waterloo, Tara Pfeiffer, Harald Huebner, Fabrizio Fierro, Regine Brox, Stefan Löber, Dorothee Weikert, Masha Y. Niv, Peter Gmeiner

Version 1 posted 24 November 2022

331

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Biological and Medicinal Chemistry

Novel Pyrazolo[3,4-c]pyridine Antagonists with Nanomolar affinity for A1 / A3 Adenosine Receptors: Binding Kinetics and Exploration of their Binding Profile Using Mutagenesis Experiments, MD simulations and TI/MD calculations

Margarita Stampelou, Anna Suchankova, Efpraxia Tzortzini, Lakshiv Dhingra, Kerry Barkan, Nikolaos Lougiakis, Panagiotis Marakos, Nikole Pouli, Graham Ladds, Antonios Kolocouris

Version 4 posted 24 November 2021

436

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Organic Chemistry

Optical Control of Cannabinoid Receptor 2–Mediated Ca2+ Release Enabled By Synthesis of Photoswitchable Probes

Roman Sarott, Alexander E.G. Viray, Patrick Pfaff, Anastasiia Sadybekov, Gabriela Rajic, Vsevolod Katritch, Erick Carreira, James Frank

Version 1 posted 28 July 2020

832

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Biological and Medicinal Chemistry

Discovery and development of macrocyclic peptide modulators of the cannabinoid 2 receptor

Natasa Tomasevic, Fabiola Susanna Emser, Jasmin Gattringer, Simon Hasinger, Roland Hellinger, Peter Keov, Manuel Felkl, Jürg Gertsch, Christian Becker, Christian Werner Gruber

Version 1 posted 14 February 2024

336

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Biological and Medicinal Chemistry

Structure-guided discovery of orexin receptor-binding PET ligands

Katharina Distler, Simone Maschauer, Eduard Neu, Harald Hübner, Jürgen Einsiedel, Olaf Prante, Peter Gmeiner

Version 1 posted 06 May 2024

83

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